BDBM50135346 4-Methyl-2-(2,4,6-trimethyl-phenylamino)-thiazole-5-carboxylic acid cyclopropylmethyl-propyl-amide::CHEMBL340469

SMILES CCCN(CC1CC1)C(=O)c1sc(Nc2c(C)cc(C)cc2C)nc1C

InChI Key InChIKey=IAWDLGWSEFUVRL-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50135346   

TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135346(4-Methyl-2-(2,4,6-trimethyl-phenylamino)-thiazole-...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity by displacement of [125I]Tyr-o-CRF from human corticotropin releasing factor receptor 1 expressed in IMR-32 human neuroblastoma cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed