BDBM50134870 4-(3-Ethyl-3H-1,2,3,5,7-pentaaza-cyclopenta[b]naphthalen-8-yl)-piperazine-1-carboxylic acid (4-phenoxy-phenyl)-amide::CHEMBL144390

SMILES CCn1nnc2cc3c(ncnc3cc12)N1CCN(CC1)C(=O)Nc1ccc(Oc2ccccc2)cc1

InChI Key InChIKey=FZLKPHLTQNXTDH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50134870   

TargetPlatelet-derived growth factor receptor beta(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50134870(4-(3-Ethyl-3H-1,2,3,5,7-pentaaza-cyclopenta[b]naph...)
Affinity DataIC50: 290nMAssay Description:Inhibition of platelet-derived growth factor receptor beta phosphorylation was measured in intact cells using a two-site enzyme linked immunosorbent ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed