BDBM50130886 CHEMBL437288::alpha-FITC-Gly(Pip)-Pro-Gly(PipAm)-Arg-Pro-Tyr--tBuGly-Leu-OH

SMILES CC(C)CC(NC(=O)C(NC(=O)C(Cc1ccc(O)cc1)NC(=O)C1CCCN1C(=O)C(CCCNC(N)=N)NC(=O)C(NC(=O)C1CCCN1C(=O)[C@@H](NC(=O)C1OC2(C3C=CC(=O)CC3Oc3cc(O)ccc23)c2ccc(NC(N)=S)cc12)C1CCNCC1)C1CCC(CC1)C(N)=N)C(C)(C)C)C(O)=O

InChI Key InChIKey=MBGDSGXTFLXGMM-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50130886   

TargetNeurotensin receptor type 1(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50130886(alpha-FITC-Gly(Pip)-Pro-Gly(PipAm)-Arg-Pro-Tyr--tB...)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity towards neurotensin receptor in membranes prepared from HT-29 cell line, relative to [111In]-labeled neurotensin peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed