BDBM50128314 CHEMBL55108::N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-benzamide

SMILES CCc1ccc(cc1)C(=O)NC1(CCCCC1)C(=O)c1cc(C)cc(C)c1

InChI Key InChIKey=MPAAOUUFYCEANT-UHFFFAOYSA-N

Data  5 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50128314   

TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  1.51E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed