BDBM50123943 CHEMBL413177::c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2

SMILES CC(C)[C@H](NC(=O)[C@@H](NC(=O)[C@H]1CCC(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc3ccccc3c2)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N1)C(C)C)C(=O)NCC(N)=O

InChI Key InChIKey=GGSUFYTUNNJUSG-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50123943   

TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonistic activity towards Melanocortin 1 receptor in Xenopus frog skin using competitive binding in the presence of 500 pM of alpha-melanocyte st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50123943(c[Pro-D-Nal(2')-Arg-Trp-Glu]-Val-Val-Gly-NH2 | CHE...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity towards Melanocortin 1 receptor in the Xenopus frog skin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed