BDBM50112771 (+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-cyclopentyl]-amide::(R,R) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-cyclopentyl]-amide::CHEMBL63417

SMILES CC(C)S(=O)(=O)N[C@@H]1CCC[C@@H]1c1ccc(Br)cc1

InChI Key InChIKey=PCKHNNAQTBNCBG-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50112771   

TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  68nMAssay Description:Potentiation of responses mediated by 100 uM L-glutamate in transfected HEK293 cells expressing human homomeric iGluR4 flip receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor 4(Human)
Nps Allelix

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  520nMAssay Description:Inhibition of GluR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetGlutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50112771((+/-) Propane-2-sulfonic acid [2-(4-bromo-phenyl)-...)
Affinity DataEC50:  520nMAssay Description:Agonist activity at GluR2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed