BDBM50096349 CHEBI:52649::CHEMBL1742484

SMILES CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](O)COP(O)(=O)OC[C@H](N)C(O)=O

InChI Key InChIKey=JZWNYZVVZXZRRH-UHFFFAOYSA-N

Data  28 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 28 hits for monomerid = 50096349   

TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  22nMAssay Description:Agonist activity at N-terminal FLAG-tagged human LPS2/P2Y10 A163F mutant transfected in HEK293-A cells co-transfected with AP-TGFalpha assessed as AP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  13nMAssay Description:Agonist activity at N-terminal FLAG-tagged human LPS2/P2Y10 V159F mutant transfected in HEK293-A cells co-transfected with AP-TGFalpha assessed as AP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  234nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  230nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Zebrafish)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Zebrafish)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at zebrafish GPR34 type b expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Zebrafish)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  129nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Zebrafish)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  130nMAssay Description:Agonist activity at zebrafish GPR34 type a expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  550nMAssay Description:Agonist activity at GPR34 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  245nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  420nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  417nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  240nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293A cells cotransfected with chimeric Galphaq/il after 1.5 hrs by alkaline phosphatase tagged-TGFalp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  520nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  550nMAssay Description:Agonist activity at GPR34 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 174(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  525nMAssay Description:Agonist activity at GPR174 (unknown origin) transfected in HEK293FT cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed
TargetPutative P2Y purinoceptor 10(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2016
Entry Details Article
PubMed