BDBM50092381 1-[7-Bromo-1-(3H-imidazol-4-ylmethyl)-3-naphthalen-1-ylmethyl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-ethanone::CHEMBL331654

SMILES CC(=O)N1Cc2cc(Br)ccc2N(Cc2cnc[nH]2)CC1Cc1cccc2ccccc12

InChI Key InChIKey=GNEPJAOLPFUJSS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50092381   

TargetDimer of Protein farnesyltransferase subunit beta(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50092381(1-[7-Bromo-1-(3H-imidazol-4-ylmethyl)-3-naphthalen...)
Affinity DataIC50: 54.5nMAssay Description:Inhibition of purified recombinant human farnesyltransferase (FT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed