BDBM50090618 CHEMBL3581733
SMILES Fc1ccc(NC(=O)N2CCc3cc(cc(N4CCCC4=O)c23)S(=O)(=O)Nc2ccc(F)cc2F)cc1
InChI Key InChIKey=LOMJQLZSGZAKFT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50090618
TargetAlpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Human)
Takeda Pharmaceutical
Curated by ChEMBL
Takeda Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of full length human MGAT2 transfected in FreeStyle293 cells assessed as dioleoylglycerol by RapidFire/MS assayMore data for this Ligand-Target Pair