BDBM50083920 3-Thiophen-2-yl-10H-benzo[4,5]imidazo[2,1-c][1,2,4]triazin-4-one::CHEMBL269112

SMILES O=c1c(n[nH]c2nc3ccccc3n12)-c1cccs1

InChI Key InChIKey=LCQXIVRCYBREJN-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50083920   

TargetAdenosine receptor A1(Bovine)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50083920(3-Thiophen-2-yl-10H-benzo[4,5]imidazo[2,1-c][1,2,4...)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptors was determined in bovine cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50083920(3-Thiophen-2-yl-10H-benzo[4,5]imidazo[2,1-c][1,2,4...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2a receptor of bovine striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed