BDBM50074552 Bis-[3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)propyl(ethyl)dimethylammonium] dibromide::CHEMBL353262

SMILES C[N+](C)(CCCN1C(=O)c2ccccc2C1=O)CCC[N+](C)(C)CCCN1C(=O)c2ccccc2C1=O

InChI Key InChIKey=MNALTKOUPBIXQI-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50074552   

TargetMuscarinic acetylcholine receptor M2(Pig)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50074552(Bis-[3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  3.80E+3nMAssay Description:Allosteric potency against the dissociation of radioligand [3H]N-methylscopolamine from the porcine cardiac Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50074552(Bis-[3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  3.80E+3nMAssay Description:Ability to dissociate radioligand [3H]NMS from muscarinic acetylcholine receptor M2 of porcine heartMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed