BDBM50074411 (2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrimidin-2-yl)-ethyl-amine::CHEMBL46479

SMILES CCN(c1nc(C)cc(C)n1)c1c(Br)cc(OC)cc1OC

InChI Key InChIKey=OQFBRKSYUGLJSA-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50074411   

TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  5nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  12nMAssay Description:Binding affinity for human recombinant corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  12nMAssay Description:Inhibition of binding of the radioligand, [125 I-Tyr0]-CRF to rat cerebral cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed