BDBM50071720 1-[4-(8-Chloro-10,10-dioxo-10,11-dihydro-5H-10lambda*6*-thia-4-aza-dibenzo[a,d]cyclohepten-5-yl)-piperazin-1-yl]-2-pyridin-4-yl-ethanone::CHEMBL86103

SMILES Clc1ccc2C(N3CCN(CC3)C(=O)Cc3ccncc3)c3ncccc3CS(=O)(=O)c2c1

InChI Key InChIKey=XOJPKPAUUVFYNE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50071720   

LigandPNGBDBM50071720(1-[4-(8-Chloro-10,10-dioxo-10,11-dihydro-5H-10lamb...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro FPT potency by measuring the ability to inhibit the transfer of [3H]farnesyl from farnesyl pyrophosphate to H-Ras-CLVS.More data for this Ligand-Target Pair
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Date in BDB:
11/10/2009
Entry Details Article
PubMed