BDBM50067688 5-[1-(3,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL342190

SMILES CC1=CC(C)(C)Nc2ccc3-c4ccccc4O\C(=C/c4cc(F)cc(F)c4)c3c12

InChI Key InChIKey=PRIMITDDFBVXLX-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50067688   

TargetProgesterone receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067688(5-[1-(3,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4...)
Affinity DataEC50:  48nMAssay Description:Effective concentration (EC50) against human progesterone receptor expressed in CV-1 cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067688(5-[1-(3,5-Difluoro-phenyl)-meth-(Z)-ylidene]-2,2,4...)
Affinity DataKi:  12.6nMAssay Description:Binding affinity against human progesterone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed