BDBM50064293 CHEMBL3403673

SMILES CC(Nc1ncnc(N)c1C#N)c1nc2ccc(F)cc2c(Cl)c1-c1ccccn1

InChI Key InChIKey=MAOHFSJHSQPOIG-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50064293   

LigandPNGBDBM50064293(CHEMBL3403673)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by biochemical Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
LigandPNGBDBM50064293(CHEMBL3403673)
Affinity DataIC50: 11nMAssay Description:Inhibition of PI3Kdelta (unknown origin) assessed as inhibition of AKT phosphorylation by cell-based HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
LigandPNGBDBM50064293(CHEMBL3403673)
Affinity DataIC50: 4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by biochemical Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
LigandPNGBDBM50064293(CHEMBL3403673)
Affinity DataIC50: 250nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by biochemical Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
LigandPNGBDBM50064293(CHEMBL3403673)
Affinity DataIC50: 230nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by biochemical Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed