BDBM50063056 CHEMBL2414732

SMILES CN1CCN(CC1)\N=C\c1c(C)n(c2ccccc12)S(=O)(=O)c1ccc2ccccc2c1

InChI Key InChIKey=NRZRJLGAEIGVHZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50063056   

Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063056(CHEMBL2414732)
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063056(CHEMBL2414732)
Affinity DataIC50: 2.04E+3nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced cAMP accumulation pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed