BDBM50060684 9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxaline::CHEMBL331304

SMILES Fc1cccc2nc(N3CCNCC3)c3cccn3c12

InChI Key InChIKey=WTIHQLOVALBPDM-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50060684   

Target5-hydroxytryptamine receptor 1B(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 106nMAssay Description:Inhibition of radiolabeled [3H]-5-HT ligand binding to 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of radiolabeled [3H]GR-113808 ligand binding to 5-hydroxytryptamine 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 268nMAssay Description:Inhibition of radiolabeled [3H]-8-OH-DPAT ligand binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 761nMAssay Description:Inhibition of radiolabeled [3H]-Ketanserin ligand binding to 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of [3H]BRL-43694 binding to 5-hydroxytryptamine 3 receptor of rat cortical homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50060684(9-Fluoro-4-piperazin-1-yl-pyrrolo[1,2-a]quinoxalin...)
Affinity DataIC50: 784nMAssay Description:Inhibition of radiolabeled [3H]mesulergine ligand binding to 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed