BDBM50055993 CHEMBL3325843

SMILES CC(C)OC(=O)N1CCC(CC1)Oc1ncnc(Oc2ccc(nc2C)S(C)(=O)=O)c1F

InChI Key InChIKey=IYPWBHJICBZOMB-UHFFFAOYSA-N

Data  1 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50055993   

TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055993(CHEMBL3325843)
Affinity DataEC50:  142nMAssay Description:Inhibition of rat GPR119 activity by homogeneous time resolved fluorescence cyclase (cAMP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055993(CHEMBL3325843)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055993(CHEMBL3325843)
Affinity DataEC50:  21nMAssay Description:Inhibition of human GPR119 activity by homogeneous time resolved fluorescence cyclase (cAMP) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed