BDBM50055368 (3-Aminooxalyl-2-methyl-1-naphthalen-1-ylmethyl-1H-indol-4-yloxy)-acetic acid::CHEMBL357804

SMILES Cc1c(c2c(n1Cc3cccc4c3cccc4)cccc2OCC(=O)O)C(=O)C(=O)N

InChI Key InChIKey=OCZWKLXXLNWSDH-UHFFFAOYSA-N

Data  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50055368   

TargetPhospholipase A2, membrane associated(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055368((3-Aminooxalyl-2-methyl-1-naphthalen-1-ylmethyl-1H...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055368((3-Aminooxalyl-2-methyl-1-naphthalen-1-ylmethyl-1H...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055368((3-Aminooxalyl-2-methyl-1-naphthalen-1-ylmethyl-1H...)
Affinity DataIC50: 1.20E+3nMAssay Description:Compound was tested for inhibition of human secretory pancreatic Phospholipase A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed