BDBM50050180 4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole::CHEMBL19172

SMILES Brc1ccc(COCCCc2cnc[nH]2)cc1

InChI Key InChIKey=BVLPCBPJCFRUBA-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50050180   

TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  12.6nMAssay Description:In vitro antagonistic activity tested against Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  14nMAssay Description:In vitro antagonistic activity tested against Histamine H3 receptor on synaptosomes from rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed