BDBM50049929 CHEMBL3317686

SMILES Cn1cc(nc1CCc1cc2ncccc2c2cc(nn12)C(F)(F)F)-c1ccccc1

InChI Key InChIKey=LJVSBBFVTOXDPW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50049929   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
University of Sassari

Curated by ChEMBL

LigandBDBM50049929(CHEMBL3317686)Copy SMILESCopy InChI

Affinity DataIC50: 190nMAssay Description:Inhibition of human PDE10A (amino acids 14 to 779) using [3H]-labelled cyclic nucleotide as substrate after 1 hr b beta countingMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/26/2016
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