BDBM50044753 2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide::CHEMBL76961

SMILES CCCCCCCCNC(=O)Cc1ccc(O)c(OC)c1

InChI Key InChIKey=RRCXCIBDXPXSRA-UHFFFAOYSA-N

Data  1 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50044753   

TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandPNGBDBM50044753(2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide |...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50044753(2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide |...)
Affinity DataEC50:  77nMAssay Description:Agonist activity at rat TRPV1 expressed in CHO cells assessed as calcium uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50044753(2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide |...)
Affinity DataKi:  848nMAssay Description:Displacement of [3H]RTX from rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed