BDBM50036549 CHEMBL3353605

SMILES CCn1ncc2cc(CN(c3ncc(cc3Cl)C(F)(F)F)S(=O)(=O)c3ccc(cc3)C(O)=O)ccc12

InChI Key InChIKey=AVABLTKDQUTJKV-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50036549   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Raqualia Pharma

Curated by ChEMBL

LigandBDBM50036549(CHEMBL3353605)Copy SMILESCopy InChI

Affinity DataIC50: 46nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition of menthol induced Ca2+ influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
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