BDBM50033243 1-Methyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]-3-phenyl-4,6-dihydro-1H-pyrazolo[3,4-b][1,4]diazepin-5-one::CHEMBL120515

SMILES Cc1nc2cnccc2n1-c1ccc(cc1)C1=Nc2c(NC(=O)C1)c(nn2C)-c1ccccc1

InChI Key InChIKey=NJBWAXLBPCZGDT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50033243   

TargetPlatelet-activating factor receptor(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033243(1-Methyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50: 2.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed