BDBM50023142 1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-1-methyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-4-yl]-amide(0.2EtOAc)::CHEMBL53907

SMILES Cc1nnc2C(NC(=O)c3cc4ccccc4[nH]3)N=C(c3ccccc3F)c3ccccc3-n12

InChI Key InChIKey=OLLDQMTZEMTSCS-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50023142   

TargetCholecystokinin receptor type A(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50023142(1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-1...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]CCK from Cholecystokinin receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50023142(1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-1...)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]gastrin from guinea pig gastric glandsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed