BDBM50017336 CHEMBL3288025

SMILES C[C@H]1CN(Cc2cc(O)cc(c2)-c2cccc(Oc3ncc(F)cc3C(=O)N[C@@H]3CC[C@@H](CC3)NC(=O)c3cc(C)n(C)n3)c2)C[C@@H](C)N1

InChI Key InChIKey=IPAJHMLMONLPPL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50017336   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50017336(CHEMBL3288025)Copy SMILESCopy InChI

Affinity DataIC50: 0.0316nMAssay Description:Inhibition of human recombinant PDE4B using [3H]cAMP by packard topcount scintillation counting analysisMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/10/2015
Entry Details Article
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