BDBM50015087 2',4',6'-Trimethyl-biphenyl-4-carboxylic acid hydroxy-methyl-amide::CHEMBL65654

SMILES CN(O)C(=O)c1ccc(cc1)-c1c(C)cc(C)cc1C

InChI Key InChIKey=GMSGKDCPRDOWJK-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50015087   

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015087(CHEMBL65654 | 2',4',6'-Trimethyl-biphenyl-4-carbox...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in rat RBL-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015087(CHEMBL65654 | 2',4',6'-Trimethyl-biphenyl-4-carbox...)
Affinity DataIC50: 64nMAssay Description:Compound was tested for its in vitro inhibitory activity against RBL-1 5-LO (time dependent)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015087(CHEMBL65654 | 2',4',6'-Trimethyl-biphenyl-4-carbox...)
Affinity DataIC50: 60nMAssay Description:Logarithmic value of inhibitory concentration against 5-lipoxygenase in rat basophilic leukemia cells (RBL-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015087(CHEMBL65654 | 2',4',6'-Trimethyl-biphenyl-4-carbox...)
Affinity DataIC50: 64nMAssay Description:In vitro inhibitory activity against 5-lipoxygenase in rat basophilic leukemia cells(RBL-1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed