BDBM50011881 3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulen-2-yl]-1-morpholin-4-yl-propenone::CHEMBL286557

SMILES Cc1nnc2CN=C(c3cc(\C=C/C(=O)N4CCOCC4)sc3-n12)c1ccccc1Cl

InChI Key InChIKey=XXYRUVMJEYVQRW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50011881   

TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011881(CHEMBL286557 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 180nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed