BDBM50003627 1-(2-Trityloxy-ethyl)-piperidine-3-carboxylic acid::CHEMBL76966

SMILES OC(=O)C1CCCN(CCOC(c2ccccc2)(c2ccccc2)c2ccccc2)C1

InChI Key InChIKey=RKUFRRGGPZSUFJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50003627   

TargetSodium- and chloride-dependent GABA transporter 1(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50003627(CHEMBL76966 | 1-(2-Trityloxy-ethyl)-piperidine-3-c...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against human GABA transporter-1 (hGAT1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed