BDBM50002158 5-Fluoro-3-[4-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-1H-indole::CHEMBL338710

SMILES Fc1ccc2[nH]cc(CCCCN3CCC(=CC3)c3ccccc3)c2c1

InChI Key InChIKey=CHPQXURJLAVZHE-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50002158   

TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(CHEMBL338710 | 5-Fluoro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataIC50: 10nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(CHEMBL338710 | 5-Fluoro-3-[4-(4-phenyl-3,6-dihydro...)
Affinity DataKi:  1.60nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed