BDBM487187 5-(4-Methoxy-phenyl)-2-methyl-3-phenyl-4H-pyrazolo[1,5-a]pyrimidin-7-one::US10953012, Example 14

SMILES COc1ccc(cc1)-c1cc(=O)n2nc(C)c(-c3ccccc3)c2[nH]1

InChI Key InChIKey=CHQLXSWIWKMWSK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 487187   

TargetPAS domain-containing serine/threonine-protein kinase [879-1323](Human)
Bioenergenix

US Patent

LigandBDBM487187(5-(4-Methoxy-phenyl)-2-methyl-3-phenyl-4H-pyrazolo...)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:Table 1: One assay for purified hPASK activity utilizes the Kinase-Glo Luminescent Kinase Assay (Promega), which quantifies the amount of ATP remaini...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In Depth
Date in BDB:
9/28/2021
Entry Details
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