BDBM483879 N-methyl-1-(cis-5- (methyl(4- (trifluoromethyl)- benzyl)amino)- octahydrocyclopenta- [c]pyrrole-2- carbonyl)-1H- pyrazole-3- carboxamide::US10927105, Ex 439::US11655217, Example 439

SMILES CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)N(C)Cc1ccc(cc1)C(F)(F)F

InChI Key InChIKey=QTWYVTHREMOYNP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 483879   

TargetMonoglyceride lipase(Human)
Lundbeck La Jolla Research Center

US Patent
LigandPNGBDBM483879(US10927105, Ex 439 | N-methyl-1-(cis-5- (methyl(4-...)
Affinity DataIC50: 100nMAssay Description:Proteomes (mouse brain membrane fraction for mouse assays; human prefrontal cortex membrane fractions for human assays) (50 mL, 1.0 mg/mL total prote...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Lundbeck La Jolla Research Center

US Patent
LigandPNGBDBM483879(US10927105, Ex 439 | N-methyl-1-(cis-5- (methyl(4-...)
Affinity DataIC50: 100nMAssay Description:Proteomes (mouse brain membrane fraction for mouse assays; human prefrontal cortex membrane fractions for human assays) (50 mL, 1.0 mg/mL total prote...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
US Patent