BDBM481647 N-cyclopentyl-N-(2-fluorobenzyl)-4- ((3-methylpiperidin-1- yl)sulfonyl)benzenesulfonamide::US10913710, Compound 58

SMILES CC1CCCN(C1)S(=O)(=O)c1ccc(cc1)S(=O)(=O)N(Cc1ccccc1F)C1CCCC1

InChI Key InChIKey=HOYVLRMYIUWDMQ-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 481647   

TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
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US Patent
LigandPNGBDBM481647(N-cyclopentyl-N-(2-fluorobenzyl)-4- ((3-methylpipe...)
Affinity DataKd:  65nMAssay Description:Binding to PDEδ was validated and quantified by means of a displacement assay employing a fluorescent-tagged analog of the HMG-CoA reductase inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2021
Entry Details
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