BDBM478099 1-((3-(8-cyano-2-(methylsulfonyl)indolizin-5- yl)pyridin-4-yl)thio)cyclobutane-1-carboxylic acid::US10894038, Example 19

SMILES CS(=O)(=O)c1cc2c(ccc(-c3cnccc3SC3(CCC3)C(O)=O)n2c1)C#N

InChI Key InChIKey=GGNJARGIHZRPCI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 478099   

TargetSolute carrier family 22 member 12(Human)
Shanghai Fochon Pharmaceutical

US Patent
LigandPNGBDBM478099(1-((3-(8-cyano-2-(methylsulfonyl)indolizin-5- yl)p...)
Affinity DataIC50: 332nMAssay Description:HEK293-URAT1 cell Lines were donated by Japan Fuji Biomedical Research Institute. Negative control cell of HEK293 (MOCK cells) which was transfected ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
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