BDBM476586 US10875864, EX. 8-24

SMILES NCC1CCN(CNc2ccc3ncc(-c4cccc(OC(F)(F)F)c4)n3n2)C(=O)C1

InChI Key InChIKey=UQEFAHDCSRWQAI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 476586   

TargetSerine/threonine-protein kinase pim-1(Human)
Sumitomo Dainippon Pharma Oncology

US Patent
LigandPNGBDBM476586(US10875864, EX. 8-24)
Affinity DataIC50: 34nMAssay Description:One illustrative manner in which Pim-1 kinase activity can be determined is by quantifying the amount of ATP remaining in solution after an in vitro ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2021
Entry Details
Go to US Patent