BDBM474310 2-((3*fluoropyridin-2-yl)methyl)-N7,N7-dimethy l-8-(3-methylimidazo[1,2-a]pyridin-6-yl)-[1,2,4] triazolo[1,5-c]pyrimidine-5,7-diamine::US10858365, Compound 100
SMILES CN(C)c1nc(N)n2nc(Cc3ncccc3F)nc2c1-c1ccc2ncc(C)n2c1
InChI Key InChIKey=OOAGAXDDBFJMBM-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 474310
Affinity DataIC50: 1.20nMAssay Description:The compounds at different concentrations were incubate with hA1 membrane (from PerkinElmer) and [3H]-8-Cyclopentyl-1,3-dipropylxanthine (DPCPX) for ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
Affinity DataIC50: 11.8nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair