BDBM461930 4-(((3r, 5r, 7r)-adamantan-1-yl)methoxy)-N-(cyclopropanesulfonimidoyl)-2-fluoro-5-methoxybenzamide::US10766858, Example 18

SMILES COc1cc(C(=O)NS(=N)(=O)C2CC2)c(F)cc1OCC12CC3CC(CC(C3)C1)C2

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 461930   

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

US Patent
LigandPNGBDBM461930(4-(((3r, 5r, 7r)-adamantan-1-yl)methoxy)-N-(cyclop...)
Affinity DataIC50: 210nMAssay Description:isolated from cells that heterologously express hNav1.7 and the β1 subunit Preparation of membranes containing recombinantly expressed sodium ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2021
Entry Details
US Patent