BDBM457843 5-chloro-1-(1-(1-(4-(ethylthio)phenyl)ethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one::US10751335, Example 5
SMILES CCSc1ccc(cc1)C(C)N1CCC(CC1)n1c2ccc(Cl)cc2[nH]c1=O
InChI Key InChIKey=NSQBVMIKHXKAKK-UHFFFAOYSA-N
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 457843
Affinity DataEC50: 291nMAssay Description:A standard [35S]GTPγS binding assay in membranes prepared from CHO cells expressing the human MOR was performed in a concentration response mann...More data for this Ligand-Target Pair
Affinity DataEC50: 622nMAssay Description:he CisBio cAMP cell based assay kit that uses HTRF technology was utilized to assess MOR-mediated inhibition of cAMP. Assays were performed according...More data for this Ligand-Target Pair
Affinity DataEC50: 291nMAssay Description:A standard [35S]GTPγS binding assay in membranes prepared from CHO cells expressing the human MOR was performed in a concentration response mann...More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:A standard [35S]GTPγS binding assay in membranes prepared from CHO cells expressing the human MOR was performed in a concentration response mann...More data for this Ligand-Target Pair