BDBM444938 6-(1-(5-Fluoro-2-methoxy-4-tetradecylphenyl)-3-methylureido)-N-(pyrimidin-2-yl)pyridine-3-sulfonamide::US10668067, Example 2-11

SMILES CCCCCCCCCCCCCCc1cc(OC)c(cc1F)N(C(=O)NC)c1ccc(cn1)S(=O)(=O)Nc1ncccn1

InChI Key InChIKey=OPMVMMJOUCOUNZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 444938   

TargetSodium channel protein type 9 subunit alpha(Human)
Amgen

US Patent

LigandBDBM444938(6-(1-(5-Fluoro-2-methoxy-4-tetradecylphenyl)-3-met...)Copy SMILESCopy InChI

Affinity DataIC50: 14nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/15/2021
Entry Details
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