BDBM444893 6-((2,4'-dichloro-3'-cyano-5-methoxy-4-::US10668067, Example 1-54

SMILES CNC(=O)N(c1ccc(cn1)S(=O)(=O)Nc1ccon1)c1cc(Cl)c(cc1OC)-c1ccc(Cl)c(c1)C#N

InChI Key InChIKey=ZFDVMRDIRSAKNT-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 444893   

LigandPNGBDBM444893(US10668067, Example 1-54 | 6-((2,4'-dichloro-3'-cy...)
Affinity DataIC50: 52nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2021
Entry Details
Go to US Patent

LigandPNGBDBM444893(US10668067, Example 1-54 | 6-((2,4'-dichloro-3'-cy...)
Affinity DataIC50: 52nMAssay Description:Inhibition of human Nav1.7 by PatchXpress assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed