BDBM434931 N-cyclobutyl-N-phenethyl-4-(4- (trifluoromethoxy)phenyl)-2H- 1,2,3-triazole-2-carboxamide::US10583137, Compound 128

SMILES FC(F)(F)Oc1ccc(cc1)-c1cnn(n1)C(=O)N(CCc1ccccc1)C1CCC1

InChI Key InChIKey=AXZSASWLSVUURE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434931   

TargetDiacylglycerol lipase-alpha(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM434931(US10583137, Compound 128 | N-cyclobutyl-N-phenethy...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2020
Entry Details
Go to US Patent

TargetDiacylglycerol lipase-beta(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM434931(US10583137, Compound 128 | N-cyclobutyl-N-phenethy...)
Affinity DataIC50: 1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2020
Entry Details
Go to US Patent