BDBM431931 ((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-dihydro-pyridin-4-yl)-phenyl]-7-fluoro-indan-1-ylamino}-2,3-dihydro-furo[3,2-c]pyridin-3-yl)-acetic Acid::US10550127, Example 17

SMILES Cc1cc(cc(C)c1-c1ccc(F)c2[C@@H](CCc12)Nc1cc2OC[C@@H](CC(O)=O)c2cn1)-c1ccn(C)c(=O)c1

InChI Key InChIKey=VKKYKJSDVMCYCG-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 431931   

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM431931(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-...)
Affinity DataEC50:  12nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
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