BDBM425999 US10513514, Compound WX032::US10513514, Number 24::US10513514, Number 25::US10513514, Number 26

SMILES Cc1cccnc1N([C@@H]1CCCNC1)C(=O)c1ccc(cc1)C1=NOC(C)(C)C1(C)O

InChI Key InChIKey=HDLQJIHCLJTIRF-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 425999   

TargetProprotein convertase subtilisin/kexin type 9(Human)
Shenzhen Salubris Pharm

US Patent
LigandPNGBDBM425999(US10513514, Compound WX032 | US10513514, Number 25...)
Affinity DataIC50: 1.00E+4nMAssay Description:1. Reagent Preparation:1) Preparation of 1× AlphaLISA test buffer solution:2.5 ml of 10× AlphaLISA test buffer solution was added to 22.5 ml of Milli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
Go to US Patent

TargetProprotein convertase subtilisin/kexin type 9(Human)
Shenzhen Salubris Pharm

US Patent
LigandPNGBDBM425999(US10513514, Compound WX032 | US10513514, Number 25...)
Affinity DataIC50: 1.00E+4nMAssay Description:1. Reagent Preparation:1) Preparation of 1× AlphaLISA test buffer solution:2.5 ml of 10× AlphaLISA test buffer solution was added to 22.5 ml of Milli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
Go to US Patent

TargetProprotein convertase subtilisin/kexin type 9(Human)
Shenzhen Salubris Pharm

US Patent
LigandPNGBDBM425999(US10513514, Compound WX032 | US10513514, Number 25...)
Affinity DataIC50: 1.00E+4nMAssay Description:1. Reagent Preparation:1) Preparation of 1× AlphaLISA test buffer solution:2.5 ml of 10× AlphaLISA test buffer solution was added to 22.5 ml of Milli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
Go to US Patent