BDBM425983 US10513514, Compound WX009::US10513514, Number 8

SMILES COc1cccnc1N([C@@H]1CCCNC1)C(=O)c1ccc(cc1)C1=NOC(C)(C)C1=O

InChI Key InChIKey=CFEJNJUAGGUQKH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 425983   

TargetProprotein convertase subtilisin/kexin type 9(Human)
Shenzhen Salubris Pharm

US Patent
LigandPNGBDBM425983(US10513514, Compound WX009 | US10513514, Number 8)
Affinity DataIC50: 1.00E+4nMAssay Description:1. Reagent Preparation:1) Preparation of 1× AlphaLISA test buffer solution:2.5 ml of 10× AlphaLISA test buffer solution was added to 22.5 ml of Milli...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2020
Entry Details
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