BDBM412919 US10399991, Example 36::US10822345, Ex 36

SMILES Cc1noc2c(C)c3[nH]c(=O)c(C)c(-c4ccccc4)c3cc12

InChI Key InChIKey=LZECURYHHUKWSL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 412919   

LigandPNGBDBM412919(US10399991, Example 36 | US10822345, Ex 36)
Affinity DataIC50: 500nMAssay Description:For a description of a Kv1.3 patch-clamp assay, see Grissmer et al., Mol. Pharmacol. 1994, 45, 1227; whole cell patch-clamp recording was performed w...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
7/27/2020
Entry Details
Go to US Patent

LigandPNGBDBM412919(US10399991, Example 36 | US10822345, Ex 36)
Affinity DataIC50: 500nMAssay Description:For a description of a Kv1.3 patch-clamp assay, see Grissmer et al., Mol. Pharmacol. 1994, 45, 1227More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/21/2021
Entry Details
Go to US Patent