BDBM412450 N-(5-(2-chloro-5-(1,5-dimethyl-1H- pyrazol-4-yl)phenyl)pyrazin-2-yl)-4- methylnicotinamide::US10399967, Compound 80

SMILES Cc1c(cnn1C)-c1ccc(Cl)c(c1)-c1cnc(NC(=O)c2cnccc2C)cn1

InChI Key InChIKey=PCXYUPSGVYKBSA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412450   

TargetInterleukin-2(Human)
Prcl Research

US Patent
LigandPNGBDBM412450(US10399967, Compound 80 | N-(5-(2-chloro-5-(1,5-di...)
Affinity DataIC50: 26nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand InfoSimilars
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Date in BDB:
7/27/2020
Entry Details
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