BDBM412378 N-(5-(2-ethyl-5-(1-methyl-1H- pyrazol-4-yl)phenyl)pyrazin-2-yl)-4- methylnicotinamide::US10399967, Compound 8

SMILES CCc1ccc(cc1-c1cnc(NC(=O)c2cnccc2C)cn1)-c1cnn(C)c1

InChI Key InChIKey=MEIKAEQFZADYSI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412378   

TargetInterleukin-2(Human)
Prcl Research

US Patent
LigandPNGBDBM412378(US10399967, Compound 8 | N-(5-(2-ethyl-5-(1-methyl...)
Affinity DataIC50: 25nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand InfoSimilars
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Date in BDB:
7/27/2020
Entry Details
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