BDBM404443 (R)-N-(1-cyanopyrrolidin- 3-yl)-5-(4-methoxyphenyl)- 1H-pyrazole-3-carboxamide::US10343992, Example 95

SMILES COc1ccc(cc1)C1C=C(NC(=O)c2ccc(cc2F)-c2cnn(C)c2)N=N1

InChI Key InChIKey=OLYNTWBALIPFSW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 404443   

TargetUbiquitin carboxyl-terminal hydrolase 30(Human)
Missions Therapeutics

US Patent
LigandPNGBDBM404443((R)-N-(1-cyanopyrrolidin- 3-yl)-5-(4-methoxyphenyl...)
Affinity DataIC50: 100nMAssay Description:Dilution plates were prepared at 21 times the final concentration (2100 μM for a final concentration of 100 μM) in 50% DMSO in a 96-well po...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2020
Entry Details
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