BDBM396633 3-[5-Chloro-2-(naphthalen-2-yloxy)-phenoxy]-azetidine::US9981909, Example 260

SMILES Clc1ccc(Oc2ccc3ccccc3c2)c(OC2CNC2)c1

InChI Key InChIKey=LWCLSZKBYNKIKU-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 396633   

TargetSodium-dependent serotonin transporter(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM396633(US9981909, Example 260 | 3-[5-Chloro-2-(naphthalen...)
Affinity DataKi:  2nMAssay Description:Receptor binding was performed using membrane fractions prepared from the HEK-293 cell line recombinantly expressing rat 5-HT7 receptors (NCBI access...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 7(Rat)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM396633(US9981909, Example 260 | 3-[5-Chloro-2-(naphthalen...)
Affinity DataKi:  16nMAssay Description:Receptor binding was performed using membrane fractions prepared from the HEK-293 cell line recombinantly expressing rat 5-HT7 receptors (NCBI access...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent