BDBM39426 7-amino-3-phenyl-6-pyrazolo[1,5-a]pyrimidinecarboxylic acid ethyl ester::7-amino-3-phenyl-pyrazolo[1,5-a]pyrimidine-6-carboxylic acid ethyl ester::MLS000075211::SMR000014414::cid_649053::ethyl 7-amino-3-phenylpyrazolo[1,5-a]pyrimidine-6-carboxylate::ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-6-carboxylate

SMILES CCOC(=O)c1cnc2c(cnn2c1N)-c1ccccc1

InChI Key InChIKey=JWQRMNHUGKWBQW-UHFFFAOYSA-N

Data  5 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 39426   

TargetSteroidogenic factor 1(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM39426(ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-...)
Affinity DataEC50:  183nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2011
Entry Details
PCBioAssay
TargetIsoform 2 of Nuclear receptor ROR-alpha (Alpha-2)(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM39426(ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-...)
Affinity DataEC50:  356nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2011
Entry Details
PCBioAssay
TargetSignal transducer and activator of transcription 3 [702-738,740-752](Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM39426(ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-...)
Affinity DataEC50: >5.57E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute (TSRI) Assay...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2011
Entry Details
PCBioAssay
TargetTranscription factor p65(Human)
Srmlsc

Curated by PubChem BioAssay
LigandPNGBDBM39426(ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-...)
Affinity DataEC50:  5.18E+3nMAssay Description:Southern Research Molecular Libraries Screening Center (SRMLSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Libraries Screening C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2011
Entry Details
PCBioAssay
TargetTumor necrosis factor receptor superfamily member 10B(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM39426(ethyl 7-azanyl-3-phenyl-pyrazolo[1,5-a]pyrimidine-...)
Affinity DataEC50: >1.25E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2013
Entry Details
PCBioAssay